GAT100 is a potent and covalent negative allosteric modulator (NAM). GAT-100 behaved as a robust positive allosteric modulator of binding of orthosteric agonist CP55,940. This novel covalent probe can serve as a useful tool for characterizing CB1R allosteric ligand-binding motifs.
Molecular Weight:
432.58
CAS Number:
[1663564-42-8]
Formula:
C25H28N4OS
Target:
Others
T70301
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