EST64454 is a sigma1 receptor (sigma1R) antagonist clinical candidate for the treatment of pain. EST64454 shows an outstanding aqueous solubility, which together with its high permeability in Caco-2 cells will allow its classification as a BCS class I compound. It also shows high metabolic stability.
Molecular Weight:
364.39
CAS Number:
[1351438-26-0]
Formula:
C18H22F2N4O2
Target:
Others|||Sigma receptor
T70908
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