()-C3001a is the racemic mixture of C3001a (CAS: 2415154-29-7). C3001a is a selective activator of the TREK channel within the two-pore-domain potassium channel (K2P) family. C3001a specifically binds to a cryptic site formed by P1 and TM4 in TREK-1, thereby promoting the selective regulation of TREK-1 activity. C3001a targets TREK channels in the peripheral nervous system, reducing the excitability of pain-sensing neurons.
Molecular Weight:
380.46
Purity:
99.13%
CAS Number:
[1374325-56-0]
Formula:
C21H20N2O3S
Target:
Others|||Potassium Channel
T71955
T71955
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