Cavalpha2delta1&NET-IN-3 (example 216) is an inhibitor targeting both the alpha2delta subunit of voltage-gated calcium channels (VGCC) and the noradrenaline transporter (NET), exhibiting inhibitory constants (Ki) ranging from 100 to 500 nM for the human alpha2delta-1 subunit of the Cav2.2 calcium channel and NET, respectively.
Molecular Weight:
466.6
CAS Number:
[2143584-82-9]
Formula:
C24H30N6O2S
Target:
Others|||Calcium Channel
T72701
* VAT and and shipping costs not included. Errors and price changes excepted