XY-06-007, a potent and selective bump-and-hole (B&H) PROTAC BRD4 BD1 L94V degrader, exhibits a DC50, 6 h of 10 nM specifically against BRD4 BD1 L94V without degrading off-targets. It also demonstrates favorable pharmacokinetics for in vivo studies [1].
Molecular Weight:
809.27
CAS Number:
[2757045-94-4]
Formula:
C41H41ClN8O8
Target:
PROTACs|||Epigenetic Reader Domain|||Others
T74380
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