Elabela(19-32) TFA, an effective fragment of ELABELA (ELA), selectively engages with the apelin receptor (APJ). This compound initiates G alphai1 and beta-arrestin-2 signaling, demonstrating EC50 values of 8.6 nM and 166 nM, respectively. It facilitates receptor internalization, lowers arterial pressure, and has a positive inotropic impact on cardiac function [1].
Molecular Weight:
1821.05
Formula:
C77H120F3N25O19S2
Target:
Apelin receptor|||Arrestin
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