I-287 is a selective, orally active PAR2 inhibitor that functions as a negative allosteric modulator of Galphaq and Galpha12/13 activity and their downstream effectors. It has been shown to attenuate Complete Freunds adjuvant-induced inflammation in mice, suggesting its utility in inflammation/immunology research [1].
Molecular Weight:
565.04
CAS Number:
[2014368-93-3]
Formula:
C30H30ClFN4O4
Target:
Protease-activated Receptor|||Others|||ERK
T78672
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