Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR partial agonism and may reduce opioid-misuse liability through D3R antagonism [1].
Molecular Weight:
410.98
Formula:
C25H31ClN2O
Target:
Dopamine Receptor|||Opioid Receptor
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