MOZ-IN-3 (Compound 6j), a potent KAT6A (MOZ) acetyltransferase inhibitor with an IC50 of 30 nM, exhibits antitumor activity against multiple myeloid leukemia cell lines, including HL-60, U937, SKNO-1, and K562. This compound also demonstrates favorable metabolic stability and pharmacokinetics [1].
Molecular Weight:
344.36
Formula:
C17H13FN2O3S
Target:
Histone Acetyltransferase
* VAT and and shipping costs not included. Errors and price changes excepted