SETD7-IN-1 (compound 7), a PFI-2 analogue, acts as both a substrate and inhibitor of histone lysine methyltransferase SETD7, exhibiting an inhibitory concentration (IC50) of 0.96 0.10 µM [1].
Target:
Histone Methyltransferase
* VAT and and shipping costs not included. Errors and price changes excepted