GA32 (compound 58r) is a potent androgen receptor (AR)/glucocorticoid receptor (GR) dual inhibitor with IC50 values of 0.13 µM and 0.83 µM for AR and GR, respectively. GA32 inhibits the proliferation of Enzalutamide-resistant, castration-resistant prostate cancer both in vitro and in vivo [1].
Molecular Weight:
417.48
CAS Number:
[1386811-71-7]
Formula:
C23H19N3O3S
Target:
Glucocorticoid Receptor|||Androgen Receptor
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