GW549390X is a dual inhibitor targeting both Fluc and VEGFR2, with IC50 values of 0.26 µM and 1.2 µM, respectively. This compound binds to the ATP pocket of FLuc via the aniline side chain, functioning as an ATP-competitive inhibitor of Fluc. It serves as a protein kinase inhibitor across ATP-dependent and -independent luciferases, potentially affecting Fluc reporter assays [1].
Molecular Weight:
236.27
CAS Number:
[135307-33-4]
Formula:
C15H12N2O
Target:
Others|||VEGFR
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