LLK203 is a potent dual-target inhibitor of USP2/USP8 with IC50 values of 0.89 µM and 0.52 µM, respectively. It promotes ERalpha degradation and induces apoptosis in breast cancer MCF-7 cells, demonstrating antitumor activity in the 4T1 tumor mice model [1].
Molecular Weight:
561.69
CAS Number:
[2758090-62-7]
Formula:
C28H23N3O4S3
Target:
DUB|||Apoptosis
T86816
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