RGH-122 (compound 43), characterized as an orally active, potent, and selective hV1a receptor antagonist, demonstrates significant affinity with a K i value of 0.3 nM and an IC 50 of 0.9 nM. It exhibits microsomal stability, indicated by a CL int value of 13/28/25 µL/min/mg [1].
Molecular Weight:
452.93
CAS Number:
[2355304-05-9]
Formula:
C24H25ClN4O3
Target:
Vasopressin Receptor
T87318
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