RWJ52353 hydrochloride, CAS [[245744-13-2]] Preis auf Anfrage

Product Overview

• Article Name: RWJ52353 hydrochloride, CAS [[245744-13-2]] Preis auf Anfrage
• Biozol Catalog Number: TGM-T87348
• Supplier Catalog Number: T87348
• Alternative Catalog Number: TGM-T87348-10MG,TGM-T87348-50MG
• Manufacturer: TargetMol
• Category: Biochemikalien

Product Description

RWJ-52353 hydrochloride is a potent oral agonist of the alpha2D adrenergic receptor (Ki: 1.5 nM) with potential analgesic properties. It exhibits pain-relief activity in abdominal tests on rats and mice and reduces agitation in mice during the hot plate and tail flick tests. Furthermore, RWJ-52353 hydrochloride modulates the organic cation transporter (OCT) subtypes by inhibiting rOCT1 and rOCT2 with IC50 values of 100 µM and 20 µM, respectively, and activating rOCT3, influencing the transport of [3H]-1-methyl-4-phenylpyridinium ([3H]MPP) in cells [1] [2].

Product Properties

• Molecular Weight: 238.73
• CAS Number: [245744-13-2]
• Formula: C11H11ClN2S
• Target: Adrenergic Receptor

Images

T87348