GS-9770, an orally active HIV protease inhibitor, demonstrates a K i of 0.16 nM. It shows potent antiviral activity against both HIV-1 and HIV-2 strains, with EC 50 values ranging from 1.9 to 26 nM. GS-9770 is metabolically stable in human liver microsomes and displays favorable pharmacokinetic properties in Sprague Dawley rats.
Molecular Weight:
811.15
CAS Number:
[2306328-43-6]
Formula:
C35H34ClF7N10O3
Target:
HIV Protease
T88206
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