Selective PAR2 peptide antagonist. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in isolated cardiac fibroblasts. Also reduces symptoms in a mouse model of dermatophyte-associated itch.
Molecular Weight:
796.97
CAS Number:
[245329-02-6]
Formula:
C39H60N10O8
Target:
Protease-activated Receptor
TP1904
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