Potent, metabolically stable neurotensin receptor agonist peptide (IC50 = 0.15 nM for inhibition of [125I]-NT binding to neonatal mouse brain, EC50 = 1.9 nM for contraction of guinea pig ileum). Produces long-lasting hypothermic, neuroprotective and analgesic effects in mice following central administration in vivo.
Molecular Weight:
746.96
CAS Number:
[139026-66-7]
Formula:
C38H66N8O7
Target:
Neurotensin Receptor
TP2012
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