High affinity apelin receptor agonist. Binds apelin receptors in left ventricle from normal and pulmonary arterial hypertensive (PAH) hearts (pKi values are 9.31 and 9.46, respectively). Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulates beta-arrestin recruitment in vitro.
Molecular Weight:
2587.12
CAS Number:
[2245073-05-4]
Formula:
C112H184N40O25S3
Target:
Apelin receptor|||Arrestin
TP2096
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