ERB 041 is a potent ERbeta agonist, displays >200-fold selectivity for ERbeta over ERalpha (IC50 values are 5 and 1216 nM for human ERbeta and ERalpha, 3.1 and 620 nM for rat ERbeta and ERalpha, and 3.7 and 750 nM for mouse ERbeta and ERalpha respectively). Pfizer Compound
Molecular Weight:
271.24
CAS Number:
[524684-52-4]
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