Reversible cell permeable p300/CBP histone acetyltransferase (HAT) inhibitor. Specific inhibition to p300 (86%) compared to N-acetyltransferase, PCAF, GCN5, Rtt109, Sas or MOZ histone acetyltransferases (<10%). Cell growth inhibitor in melanoma and non-small-cell-lung (NSCL) human cancer cell lines. Synonyms: (E)-4-(4-((5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl)-methylene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid CAS Number: 328968-36-1 Molecular Weight: 445.4 Molecular Formula: C24H19N3O6 Solubility: DMSO (10mg/ml). Appearance: Supplied as a red solid. Purity: 98% (NMR) Storage and Stability: Store at -20C under inert atmosphere. For maximum recovery of product, centrifuge the original vial prior to removing the cap.
Molecular Weight:
445.4
Purity:
98% (NMR)
Form:
Supplied as a red solid.
CAS Number:
[328968-36-1]
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