Ghrelin receptor antagonist (GHS-R1a) (Ki = 17nM). Displays no significant affinity for the motilin receptor (Ki = 6uM). Blocks the effects of ghrelin on insulin secretion both in vivo and in vitro. Improves glucose homeostasis in vivo. Purity: 98% Solubility: Soluble to 100mM in DMSO and to 100mM in water Storage: Desiccate at RT Alternate Name: 6-(4-Fluorophenoxy)-2-methyl-3-[[(3S)-1-(1-methylethyl)-3-piperidinyl]methyl]-4(3H)-quinazolinone CAS Number: 875258-85-8 Molecular Formula: C24H28FN3O2.HCl Molecular Weight: 445.96 Storage: -20C
Molecular Weight:
445.96
Purity:
98% (HPLC)
Form:
Supplied as a tan solid.
CAS Number:
[875258-85-8]
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