GYKI 52466 Hydrochloride (1-(4-Aminophenyl)-4-methyl-7,8-methylenedioxy-5H-2,3-benzodiazepine Hydrochloride, GYKI-52,466, GYK I52466), CAS [[102771-26-6]]

Product Overview

• Article Name: GYKI 52466 Hydrochloride (1-(4-Aminophenyl)-4-methyl-7,8-methylenedioxy-5H-2,3-benzodiazepine Hydrochloride, GYKI-52,466, GYK I52466), CAS [[102771-26-6]]
• Biozol Catalog Number: USB-217409
• Supplier Catalog Number: 217409
• Alternative Catalog Number: USB-217409-10
• Manufacturer: US Biological
• Category: Biochemikalien

Product Description

A potent negative allosteric modulator selective for AMPA glutamate receptors (IC50 = 10-20uM) over kainate (IC50 ~450uM) and nMDA (IC50 >> 50uM) receptors. Commonly used as neuroprotectant, anticonvulsant, and skeletal muscle relaxant. Biologically viable admitted orally or systematically. CAS Number: 102771-26-6 Formula: C17H15N3O2HCl Primary Target: AMPA Primary Target IC50: 10-20 M Molar Mass: 329.78 Solubility: H2O Storage and Stability: May be stored at 4C. For long-term storage, aliquot and store at 4C. Do not freeze. For maximum recovery of product, centrifuge the original vial prior to removing the cap. Further dilutions can be made in assay buffer.

Product Properties

• Molecular Weight: 329.78
• Purity: ~98% (HPLC)
• Form: Supplied as a yellow solid.
• CAS Number: [102771-26-6]