SR95531 (Gabazine) Hydrobromide, CAS [[104104-50-9]]

Product Overview

• Article Name: SR95531 (Gabazine) Hydrobromide, CAS [[104104-50-9]]
• Biozol Catalog Number: USB-217808
• Supplier Catalog Number: 217808
• Alternative Catalog Number: USB-217808-10,USB-217808-25,USB-217808-50
• Manufacturer: US Biological
• Category: Biochemikalien

Product Description

A selective, competitive antagonist of GABAA receptor (IC50 = 440nM) that does not affect pentobarbitone or etomidate- induced currents even at high concentrations (~100uM). Also shown to block glycine receptors, but with low affinity (Kb = 190uM). Synonyms: Gabazine, GABAA Receptor Antagonist, SR-95531, 6-imino-3-(4-methoxyphenyl)-1(6H)-pyridazinebutanoic acid, monohydrobromide CAS No: 104104-50-9 Molecular Formula: C15H17N3O3 HBr Molecular Weight: 368.23 Appearance: White solid Purity: 98% (HPLC) Primary Target: GABA-A Primary Target IC50: 440nM Proton NMR: Conforms to structure Elemental Analysis: C% :47.50-50.50% H%: 4.00-6.00% N%: 10.00-13.00% Water Molecules: 1.0mol Solubility: Water (25mM), MeOH:PBS (pH 7.2), (1:1): 0.5mg/ml, Methanol: 1mg/ml Storage and Stability: Lyophilized powder may be stored at 4C Do not freeze. Stable for 6 months after receipt at 4C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.

Product Properties

• Molecular Weight: 368.23
• Purity: 98% (HPLC)
• Form: White solid
• CAS Number: [104104-50-9]