Potent and selective 5-HT2C agonist (IC50 values are 12 and 633 nM for 5-HT2C and 5-HT2A receptors respectively). Displays high affinity for the 5-HT2B receptor (Ki = 38 nM) but acts as an inverse agonist. Active in vivo, inhibits scratching in a mouse model of OCD. Synonyms: 3-[2-(Dimethylamino)ethyl]-1-methylindol-4-ol CAS Number: 1465-16-3 Molecular Weight: 218.29 Molecular Formula: C13H18N2O Solubility: DMSO to 100mM, ethanol to 10mM Method for Determining Identity: Proton NMR and Mass Spectrometric analysis Melting Point: 125-127C Appearance: Supplied as a brown solid. Purity: 99% (HPLC) Storage and Stability: Store at 4C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.
Molecular Weight:
218.29
Purity:
99% (HPLC)
Form:
Supplied as a brown solid.
CAS Number:
[1465-16-3]
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