LY2183240 is is a potent inhibitor of FAAH activity, and the uptake and enzymatic hydrolysis of anandamide. Potent, covalent inhibitor of the EC-degrading enzyme fatty acid amide hydrolase (FAAH). Disrupts the cellular uptake of the lipid endocannabinoid (EC) anandamide and promote analgesia in vivo. LAlso an inhibitor of monoacylgylcerol lipase (MGL). Synonyms: 5-[(1,1-Biphenyl]-4-yl)methyl]-N,N-dimethyl-1H-tetrazole-1-carboxamide CAS No: 874902-19-9 Molecular Formula: C17H17N5O Molecular Weight: 307.35 Appearance: White to off-white powder Purity: 99% (HPLC) Solubility: DMF: 3mg/ml, DMSO: 2mg/ml, Ethanol: 10mg/ml, Ethanol:PBS(pH 7.2) (1:5): 0.1mg/ml Storage and Stability: May be stored at RT for short-term only. Long-term storage is recommended at -20C. For maximum recovery of product, centrifuge the original vial prior to removing the cap. Stock Solution Storage: 0-4C for short term (days to weeks), or -20C for long term (months).
Molecular Weight:
307.35
Purity:
99% (HPLC)
Form:
White to off-white powder
CAS Number:
[874902-19-9]
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