EPI-001, a selective inhibitor of Androgen Receptor (AR), targets transactivation unit 5 (Tau-5) of the AR. EPI-001 can inhibit transactivation of the AR amino-terminal domain (NTD), with an IC50 of ~6 µM. EPI-001 is also a selective modulator of PPARgamma. EPI-001 is active against castration-resistant prostate cancer[1][2][3].
Molecular Weight:
394.89
Purity:
99.34
CAS Number:
[227947-06-0]
Formula:
C21H27ClO5
Target:
Androgen Receptor,Apoptosis,PPAR
Application Notes:
Reference compound
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