CCG258208 (hydrochloride)

Product Overview

• Article Name: CCG258208 (hydrochloride)
• Biozol Catalog Number: MCE-HY-109562A
• Supplier Catalog Number: HY-109562A
• Alternative Catalog Number: MCE-HY-109562A-10MG,MCE-HY-109562A-50MG,MCE-HY-109562A-10MMX1ML,MCE-HY-109562A-25MG,MCE-HY-109562A-100MG,MCE-HY-109562A-5MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: GRK2-IN-1 (hydrochloride)

Product Description

CCG258208 (GRK2-IN-1) hydrochloride is a potent and selective GRK2 (G protein-coupled receptor kinase 2) inhibitor (IC50=30 nM) while maintaining 230-fold selectivity over GRK5 (IC50=7.09 µM) and more than 2500-fold selectivity over GRK1 (IC50=87.3 µM), PKA, and ROCK1. CCG258208 hydrochloride can be used in heart failure research[1].

Product Properties

• Molecular Weight: 488.94
• Purity: 98.05
• Formula: C24H26ClFN4O4
• Target: G Protein-coupled Receptor Kinase (GRK)

Application Notes

• Application Notes: MCE Product type: Reference compound