(E)-KN-93 phosphate is an inhibitor for Ca2+/calmodulin-dependent protein kinase II (CaMK II) with IC50 of 9 µM and 3 µM, for CaMKIIdelta monomer and CaMKIIdelta dodecamer. (E)-KN-93 phosphate binds competitively with Ca2+/CaM, and disrupts their interaction with CaMK II, and thus inhibits the CaMK II activation[1].
Molecular Weight:
599.03
Purity:
99.85
CAS Number:
[1188890-41-6]
Formula:
C26H32ClN2O8PS
Target:
CaMK
Application Notes:
MCE Product type: Reference compound1
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