BI-9321 (trihydrochloride), CAS [[2387510-87-2]]

Product Overview

• Article Name: BI-9321 (trihydrochloride), CAS [[2387510-87-2]]
• Biozol Catalog Number: MCE-HY-114208A
• Supplier Catalog Number: HY-114208A
• Alternative Catalog Number: MCE-HY-114208A-100MG,MCE-HY-114208A-10MG,MCE-HY-114208A-25MG,MCE-HY-114208A-10MMX1ML,MCE-HY-114208A-5MG,MCE-HY-114208A-50MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

BI-9321 trihydrochloride is a potent, selective and cellular active nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist with a Kd value of 166 nM. BI-9321 trihydrochloride is inactive against NSD2-PWWP1 and NSD3-PWWP2. BI-9321 trihydrochloride specifically disrupts histone interactions of the NSD3-PWWP1 domain with an IC50 of 1.2 µM in U2OS cells[1].

Product Properties

• Molecular Weight: 469.81
• Purity: 99.83
• CAS Number: [2387510-87-2]
• Formula: C22H24Cl3FN4
• Target: Histone Methyltransferase

Application Notes

• Application Notes: MCE Product type: Reference compound