PROTAC FLT-3 degrader 1, CAS [[2230826-81-8]]

Catalog Number: MCE-HY-114323
Article Name: PROTAC FLT-3 degrader 1, CAS [[2230826-81-8]]
Biozol Catalog Number: MCE-HY-114323
Supplier Catalog Number: HY-114323
Alternative Catalog Number: MCE-HY-114323-10MMX1ML,MCE-HY-114323-50MG,MCE-HY-114323-25MG,MCE-HY-114323-10MG,MCE-HY-114323-5MG,MCE-HY-114323-100MG,MCE-HY-114323-1MG
Manufacturer: MedchemExpress
Category: Biochemikalien
PROTAC FLT-3 degrader 1 is an effective and selective FLT-3 PROTAC degrader with an IC50 of 0.6 nM. PROTAC FLT-3 degrader 1 inhibits both FLT-3 and FLT-3 ITD mutants. PROTAC FLT-3 degrader 1 has the activity of anti-proliferation and induction of apoptosis, which can be used in the study of tumor. (Pink: FLT3 ligand (HY-168702), Black: Linker (HY-124380), Blue: VHL ligand (HY-125845))[1].
Molecular Weight: 1020.23
Purity: 99.74
CAS Number: [2230826-81-8]
Formula: C52H61N9O9S2
Target: Apoptosis,ERK,FLT3,MEK,PROTACs,STAT
Application Notes: Reference compound