GRPR antagonist-1, CAS [[3052544-28-9]]

Product Overview

• Article Name: GRPR antagonist-1, CAS [[3052544-28-9]]
• Biozol Catalog Number: MCE-HY-115974
• Supplier Catalog Number: HY-115974
• Alternative Catalog Number: MCE-HY-115974-100MG,MCE-HY-115974-50MG,MCE-HY-115974-25MG,MCE-HY-115974-10MG,MCE-HY-115974-5MG,MCE-HY-115974-10MMX1ML
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

GRPR antagonist-1 is a potent gastrin releasing peptide receptor (GRPR) antagonist, having the cytotoxicity against certain cancer cells (IC50 of 4.97, 4.36 and 3.40 µM in PC3, Pan02 and HGC-27 cells, respectively). GRPR antagonist-1 inhibits HGC-27 cell viability by decreasing the Bcl-2 level and increasing the Bax level, causing apoptosis, with anticancer activity[1].

Product Properties

• Molecular Weight: 558.59
• Purity: 99.80
• CAS Number: [3052544-28-9]
• Formula: C29H33F3N4O4
• Target: Bombesin Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound