Rosiglitazone maleate (BRL 49653C) is a potent and selective activator of PPARgamma, with EC50s of 30 nM, 100 nM and 60 nM for PPARgamma1, PPARgamma2, and PPARgamma, respectively, and a Kd of appr 40 nM for PPARgamma, Rosiglitazone maleate is also an modulator of TRP channels, inhibits TRP melastatin 2 (TRPM2), TRPM3 and activates TRP canonical 5 (TRPC5).
Molecular Weight:
473.50
Purity:
99.73
CAS Number:
[155141-29-0]
Formula:
C22H23N3O7S
Target:
Autophagy,Ferroptosis,PPAR,TRP Channel
Application Notes:
MCE Product type: Reference compound1
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