TRPV2-selective blocker 1 (compound IV2-1) is a selective TRPV2 channel blocker with an IC50 of 6.3 µM. TRPV2-selective blocker 1 does not affect TRPV1, TRPV3 or TRPV4 channels. TRPV2-selective blocker 1 also inhibits TRPV2-mediated Ca2+ influx in macrophages, and inhibits macrophage phagocytosis[1].
Molecular Weight:
278.43
Purity:
99.84
CAS Number:
[2242724-49-6]
Formula:
C15H18OS2
Target:
TRP Channel
Application Notes:
MCE Product type: Reference compound
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