P7-2302 inhibits PDE7 and PDE4B with IC50 of 0.18 nM and 77.3 nM. P7-2302 inhibits the efflux of P-gp and BCRP (breast cancer resistance protein), exhibits low uptake in rats brain. P7-2302 can be used as a PET tracer when labeled with 18F[1].
Molecular Weight:
462.87
Formula:
C23H21ClF2N2O4
Target:
Phosphodiesterase (PDE)
Application Notes:
MCE Product type: Reference compound
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