SCH772984 is a highly selective and ATP-competitive ERK inhibitor, with IC50s of 4 and 1 nM for ERK1 and ERK2, respectively. SCH772984 has antitumor activity in MAPK inhibitor-na ve and MAPK inhibitor-resistant cells containing BRAF or RAS mutations[1].
Molecular Weight:
587.67
Purity:
99.83
CAS Number:
[942183-80-4]
Formula:
C33H33N9O2
Target:
ERK
Application Notes:
MCE Product type: Reference compound
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