A-582941 dihydrochloride is a potent, selective and brain-penetrant partial agonist of alpha7 nAChR, with Kis of 10.8 and 16.7 nM in rat brain membranes and human frontal cortex, respectively. A-582941 dihydrochloride also binds to human 5-HT3 receptor with a Ki of 150 nM. A-582941 has the potential for cognitive deficits associated with various neurodegenerative and psychiatric disorders research[1][2].
Molecular Weight:
353.29
Purity:
99.78
CAS Number:
[848591-90-2]
Formula:
C17H22Cl2N4
Target:
5-HT Receptor,nAChR
Application Notes:
MCE Product type: Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted
