Trimipramine maleate is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively[1]. Trimipramine maleate is also a potent and selective inhibitor targeting human noradrenaline (hNAT), serotonin (hSERT) and organic cation transporters (hOCT1, hOCT2) with IC50 values of 4.99 µM, 2.11 µM, 3.72 µM, 8.00 µM, respectively[2]. Trimipramine maleate has vascular activity and anxiolytic efficacy[3].
Molecular Weight:
410.51
Purity:
99.97
CAS Number:
[521-78-8]
Formula:
C24H30N2O4
Target:
5-HT Receptor,Bacterial
Application Notes:
Reference compound
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