CXCR4 antagonist 8 (Compound 3) is a potent inhibitor of CXCR4, exhibiting an IC50 value of 57 nM in antagonism and effectively inhibiting CXCL12-induced cytosolic calcium increase with an IC50 of 0.24 nM. Additionally, Compound 3 is efficacious in inhibiting CXCL12/CXCR4-mediated cell migration [1].
Molecular Weight:
362.47
CAS Number:
[2304750-84-1]
Formula:
C21H26N6
Target:
Others|||CXCR
T61363
* VAT and and shipping costs not included. Errors and price changes excepted