HEMTAC CDK4/6 degrader 1, CAS [[2821803-61-4]]

Catalog Number: TGM-T75029
Article Name: HEMTAC CDK4/6 degrader 1, CAS [[2821803-61-4]]
Biozol Catalog Number: TGM-T75029
Supplier Catalog Number: T75029
Alternative Catalog Number: TGM-T75029-5MG
Manufacturer: TargetMol
Category: Biochemikalien
HEMTAC CDK4/6 degrader 1 is a PROTAC connected by ligands for HSP90 and CDK4/6 with a \( K_d \) value of 35.7 µM. It induces CDK4/6 degradation in B16F10 melanoma cells, arrests the cell cycle at the G0/G1 phase, and induces apoptosis. HEMTAC CDK4/6 degrader 1 can be used in cancer research [1].
Molecular Weight: 953.49
CAS Number: [2821803-61-4]
Formula: C48H53ClN16O4
Target: PROTACs|||Apoptosis|||CDK|||Others